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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2600 | AG490 | Zinc02557947,Tyrphostin AG 490,AG 490,AG-490,Tyrphostin B42 | EGFR , JAK , STAT , Autophagy |
AG490 (Tyrphostin B42) is an inhibitor of EGFR (IC50: 0.1 μM). It is 135-fold more selective for EGFR than ErbB2, also inhibits JAK2 with no effect to Lyn, Lck, Syk, Btk, and Src. |